BIA 10-2474
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BIA 10-2474 is an experimental fatty acid amide hydrolase inhibitor developed by the Portuguese pharmaceutical company Bial-Portela & Ca. SA. It interacts with the human endocannabinoid system.[1] The drug was in development for the treatment of a range of different medical conditions from anxiety disorder to Parkinson's disease, also for the treatment of chronic pain of multiple sclerosis, cancer, hypertension or the treatment of obesity.[2] A clinical trial with this drug was underway in Rennes, France, in January 2016, in which serious adverse events occurred affecting five participants, including the death of one man.[1][3][4][5] The underlying mechanism that caused the acute neurotoxicity of this molecule remains unknown.[6][7]
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Routes of administration | Oral |
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Formula | C16H20N4O2 |
Molar mass | 300.362 g·mol−1 |
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